Ethylamine → HCID 49782710, compound

Participants

Reaction Steps

As described for example 40c, 2-{2-[3-(5-fluoro-pyridin-2-yl)-5-methyl-isoxazol-4-yl]-ethyl}-thiazole-5-carboxylic acid (67 mg, 0.20 mmol) was converted, using ethylamine (2M solution in THF) instead of 4-aminotetrahydropyran, to the title compound (42 mg, 58%) which was obtained as a white solid. MS: m/e=361.2 [M+H]+.

Provenance & Evidence