HuagongsheHuagongshe Chemistry Print Report · For research reference only
Benzo[C][1,2,5]Oxadiazole-5-Boronic Acid → 4-Benzo[1,2,5]oxadiazol-5-yl-1H-indole-2-carboxylic acid [1-(2-azepan-1-yl-ethyl)-piperidin-4-yl]-amide
Participants
| Role | Name | HCID | Charge |
|---|---|---|---|
| Reactant | Benzo[C][1,2,5]Oxadiazole-5-Boronic Acid | HCID 4672597 | — |
| Reactant | 4-Bromo-1H-indole-2-carboxylic acid [1-(2-azepan-1-yl-ethyl)-piperidin-4-yl]-amide | HCID 59600248 | — |
| Product | 4-Benzo[1,2,5]oxadiazol-5-yl-1H-indole-2-carboxylic acid [1-(2-azepan-1-yl-ethyl)-piperidin-4-yl]-amide | HCID 59600240 | — |
Reaction Steps
This compound is synthesized from compound 194 (see example 156) and benzo[1,2,5]oxadiazol-5-yl-boronic acid analogously to the method described in Example 156.
Provenance & Evidence
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| Patent number | US08183366B2 |
| Source dataset | uspto-grants-2012_05 |
| ORD ID | ord-452d5b846cf64c10aa8b935e9914e53a |
| Source note | uspto-grants-2012_05 |