2-Fluorophenylboronic acid → HCID 57753225, compound

HRID 1931010Notes

Reaction equation

HRID 1931010 reaction equation
I[C:2]1[CH:10]=[CH:9][C:8]([S:11]([CH3:14])(=[O:13])=[O:12])=[CH:7][C:3]=1[C:4]([OH:6])=[O:5].[F:15][C:16]1[CH:21]=[CH:20][CH:19]=[CH:18][C:17]=1B(O)O>>[F:15][C:16]1[CH:21]=[CH:20][CH:19]=[CH:18][C:17]=1[C:2]1[C:3]([C:4]([OH:6])=[O:5])=[CH:7][C:8]([S:11]([CH3:14])(=[O:13])=[O:12])=[CH:9][CH:10]=1

Participants

3

Reactant 2

HCID 27343542-Fluorophenylboronic acidHCID 574452812-Iodo-5-methanesulfonyl-benzoic acid

Product 1

HCID 57753225HCID 57753225, compound

Procedure

Prepared in analogy to Example B25 from 2-Iodo-5-methanesulfonyl-benzoic acid (example B19(b)) and 2-fluorobenzeneboronic acid. Light brown solid.

Sources & evidence

ORD record
ord-593f7fb718ae41298b746c0c77f30c36
Source dataset
uspto-grants-2012_05
Patent number
US08188139B2

Reaction notes

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