3-Benzyloxy-phenylboronic acid → HCID 67329648, compound

HRID 1942555Notes

Reaction equation

HRID 1942555 reaction equation
FC(F)(F)S(O[C:7]1[CH2:12][CH2:11][N:10]([C:13]([O:15][C:16]([CH3:19])([CH3:18])[CH3:17])=[O:14])[CH2:9][C:8]=1[C:20]([O:22][CH2:23][CH3:24])=[O:21])(=O)=O.[CH2:27]([O:34][C:35]1[CH:36]=[C:37](B(O)O)[CH:38]=[CH:39][CH:40]=1)[C:28]1[CH:33]=[CH:32][CH:31]=[CH:30][CH:29]=1>>[CH2:27]([O:34][C:35]1[CH:40]=[C:39]([C:7]2[CH2:12][CH2:11][N:10]([C:13]([O:15][C:16]([CH3:19])([CH3:18])[CH3:17])=[O:14])[CH2:9][C:8]=2[C:20]([O:22][CH2:23][CH3:24])=[O:21])[CH:38]=[CH:37][CH:36]=1)[C:28]1[CH:33]=[CH:32][CH:31]=[CH:30][CH:29]=1

Participants

3

Reactant 2

HCID 27343133-Benzyloxy-phenylboronic acidHCID 222284091-(tert-Butyl) 3-ethyl 4-(((trifluoromethyl)sulfonyl)oxy)-5,6-dihydropyridine-1,3(2H)-dicarboxylate

Product 1

HCID 67329648HCID 67329648, compound

Procedure

Using 1-tert-butyl 3-ethyl 4-{[(trifluoromethyl)sulfonyl]oxy}-5,6-dihydropyridin-1,3(2H)-dicarboxylate and 3-benzyloxyphenylboronic acid, the title compound was obtained in a similar manner to Reference Example 550.

Sources & evidence

ORD record
ord-8a379f04f4dc46acb52458ba66247630
Source dataset
uspto-grants-2013_03
Patent number
US08389511B2

Reaction notes

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