HCID 58207875, compound → HCID 58207895, compound

HRID 1958504Notes

Reaction equation

HRID 1958504 reaction equation
Br[C:2]1[S:6][C:5]([S:7][CH:8]([CH3:10])[CH3:9])=[N:4][CH:3]=1.[C:11]1([CH3:29])[CH:16]=[CH:15][CH:14]=[CH:13][C:12]=1[C:17]1[C:18]2[N:19]([CH:26]=[CH:27][N:28]=2)[CH:20]=[C:21](B(O)O)[CH:22]=1>>[CH:8]([S:7][C:5]1[S:6][C:2]([C:21]2[CH:22]=[C:17]([C:12]3[CH:13]=[CH:14][CH:15]=[CH:16][C:11]=3[CH3:29])[C:18]3[N:19]([CH:26]=[CH:27][N:28]=3)[CH:20]=2)=[CH:3][N:4]=1)([CH3:10])[CH3:9]

Participants

3

Reactant 2

HCID 58207875HCID 58207875, compoundHCID 67008224HCID 67008224, compound

Product 1

HCID 58207895HCID 58207895, compound

Procedure

Prepared using the procedure describe for Example 34, step 4 from 5-bromo-2-(isopropylthio)thiazole and 8-o-tolylimidazo[1,2-a]pyridin-6-ylboronic acid. LCMS (Conditions C): Tr 2.96 min.; (M+H)+: 366.3.

Workup

  1. customPrepared
  2. customTr 2.96 min.

Sources & evidence

ORD record
ord-24f027e4b981477aa6713c46163c60e7
Source dataset
uspto-grants-2013_04
Patent number
US08410128B2

Reaction notes

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