tert-Butyl carbamate → HCID 59443087, compound

HRID 1959119Notes

Reaction equation

HRID 1959119 reaction equation
Cl[C:2]1[CH:11]=[C:10]2[C:5]([C:6]([C:15]3[CH:20]=[CH:19][C:18]([F:21])=[CH:17][CH:16]=3)=[C:7]([CH3:14])[C:8]([CH3:13])([CH3:12])[O:9]2)=[CH:4][CH:3]=1.[C:22](=[O:29])([O:24][C:25]([CH3:28])([CH3:27])[CH3:26])[NH2:23]>>[F:21][C:18]1[CH:19]=[CH:20][C:15]([C:6]2[C:5]3[C:10](=[CH:11][C:2]([NH:23][C:22](=[O:29])[O:24][C:25]([CH3:28])([CH3:27])[CH3:26])=[CH:3][CH:4]=3)[O:9][C:8]([CH3:13])([CH3:12])[C:7]=2[CH3:14])=[CH:16][CH:17]=1

Participants

3

Reactant 2

HCID 77922tert-Butyl carbamateHCID 59442921HCID 59442921, compound

Product 1

HCID 59443087HCID 59443087, compound

Procedure

The compound obtained in (3) described above (100 mg) and tert-butyl carbamate (125 mg) were treated in the same manner as Reference Example 5(4) to give the titled compound (126 mg) as a pale brown powder.

Sources & evidence

ORD record
ord-6ca14e9036b941b89cec1fb5b6c90a37
Source dataset
uspto-grants-2013_04
Patent number
US08410166B2

Reaction notes

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