反应详情

As described for example 4c, 5-(5-methyl-3-phenyl-isoxazol-4-ylmethoxy)-pyridine-2-carboxylic acid (100 mg, 0.32 mmol) was converted, using N-aminomorpholine instead of N,N-dimethylhydrazine, to the title compound (62 mg, 49%) which was obtained as a light yellow oil. MS: m/e=395.3 [M+H]+.