5-Chloro-2-methoxyphenylboronic acid → HCID 67241540, compound
Reaction equation
Br[C:2]1[CH:7]=[CH:6][C:5]([S:8]([C:11]2[CH:16]=[CH:15][CH:14]=[CH:13][CH:12]=2)(=[O:10])=[O:9])=[CH:4][C:3]=1[F:17].[Cl:18][C:19]1[CH:20]=[CH:21][C:22]([O:28][CH3:29])=[C:23](B(O)O)[CH:24]=1>>[C:11]1([S:8]([C:5]2[CH:6]=[CH:7][C:2]([C:21]3[CH:20]=[C:19]([Cl:18])[CH:24]=[CH:23][C:22]=3[O:28][CH3:29])=[C:3]([F:17])[CH:4]=2)(=[O:10])=[O:9])[CH:16]=[CH:15][CH:14]=[CH:13][CH:12]=1Participants
3
Procedure
The subtitle compound was prepared by the method of example 2 step (ii) using the product of example 5 step (i) and 5-chloro-2-methoxybenzene boronic acid.
Sources & evidence
- ORD record
- ord-f471f4de83b645c1bf51140586904ff8
- Source dataset
- uspto-grants-2013_04
- Patent number
- US08415394B2
Reaction notes
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