(2-Methoxy-5-methylphenyl)boronic acid → HCID 68436456, compound

HRID 1963685Notes

Reaction equation

HRID 1963685 reaction equation
Br[C:2]1[CH:7]=[CH:6][C:5]([S:8]([C:11]2[CH:16]=[CH:15][C:14]([F:17])=[CH:13][CH:12]=2)(=[O:10])=[O:9])=[C:4]([F:18])[CH:3]=1.[CH3:19][O:20][C:21]1[CH:26]=[CH:25][C:24]([CH3:27])=[CH:23][C:22]=1B(O)O>>[F:17][C:14]1[CH:15]=[CH:16][C:11]([S:8]([C:5]2[CH:6]=[CH:7][C:2]([C:22]3[CH:23]=[C:24]([CH3:27])[CH:25]=[CH:26][C:21]=3[O:20][CH3:19])=[CH:3][C:4]=2[F:18])(=[O:10])=[O:9])=[CH:12][CH:13]=1

Participants

3

Reactant 2

HCID 2773485(2-Methoxy-5-methylphenyl)boronic acidHCID 67239250HCID 67239250, compound

Product 1

HCID 68436456HCID 68436456, compound

Procedure

The subtitle compound was prepared by the method of example 2 step (ii) using the product of example 4 step (i) and (2-methoxy-5-methylphenyl)boronic acid.

Sources & evidence

ORD record
ord-4e4f1e5f1c5d4ae7911e687cd6ac327c
Source dataset
uspto-grants-2013_04
Patent number
US08415394B2

Reaction notes

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