3-(Piperidine-1-sulfonyl)benzoic acid → HCID 2952736, compound
Reaction equation
[N:1]1([S:7]([C:10]2[CH:11]=[C:12]([CH:16]=[CH:17][CH:18]=2)[C:13]([OH:15])=O)(=[O:9])=[O:8])[CH2:6][CH2:5][CH2:4][CH2:3][CH2:2]1.[NH2:19][C:20]1[CH:24]=[CH:23][O:22][N:21]=1>>[O:22]1[CH:23]=[CH:24][C:20]([NH:19][C:13](=[O:15])[C:12]2[CH:16]=[CH:17][CH:18]=[C:10]([S:7]([N:1]3[CH2:2][CH2:3][CH2:4][CH2:5][CH2:6]3)(=[O:8])=[O:9])[CH:11]=2)=[N:21]1Participants
3
Procedure
The entitled compound was produced according to the method of Example 73 but using 3-(piperidin-1-ylsulfonyl)benzoic acid and 3-aminoisoxazole as the starting materials.
Workup
- customThe entitled compound was produced
Sources & evidence
- ORD record
- ord-c63547f9562944ddae9fc21f49a60dd3
- Source dataset
- uspto-grants-2013_04
- Patent number
- US08420823B2
Reaction notes
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