3-(Piperidine-1-sulfonyl)benzoic acid → HCID 2710158, compound

HRID 1967499Notes

Reaction equation

HRID 1967499 reaction equation
[N:1]1([S:7]([C:10]2[CH:11]=[C:12]([CH:16]=[CH:17][CH:18]=2)[C:13]([OH:15])=O)(=[O:9])=[O:8])[CH2:6][CH2:5][CH2:4][CH2:3][CH2:2]1.[C@@H:19]1([NH2:29])[C:28]2[C:23](=[CH:24][CH:25]=[CH:26][CH:27]=2)[CH2:22][CH2:21][CH2:20]1>>[N:1]1([S:7]([C:10]2[CH:11]=[C:12]([CH:16]=[CH:17][CH:18]=2)[C:13]([NH:29][C@@H:19]2[C:28]3[C:23](=[CH:24][CH:25]=[CH:26][CH:27]=3)[CH2:22][CH2:21][CH2:20]2)=[O:15])(=[O:8])=[O:9])[CH2:2][CH2:3][CH2:4][CH2:5][CH2:6]1

Participants

3

Reactant 2

HCID 7678893-(Piperidine-1-sulfonyl)benzoic acidHCID 70580741-Aminotetralin, (S)-

Product 1

HCID 2710158HCID 2710158, compound

Procedure

The entitled compound was produced according to the method of Example 73 but using 3-(piperidin-1-ylsulfonyl)benzoic acid and (S)-(+)-1,2,3,4-tetrahydro-1-naphthylamine as the starting materials.

Workup

  1. customThe entitled compound was produced

Sources & evidence

ORD record
ord-af0d29f9a8b349e7a0502220ca8c593a
Source dataset
uspto-grants-2013_04
Patent number
US08420823B2

Reaction notes

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