3-(Piperidine-1-sulfonyl)benzoic acid → N-(3-methoxypyridin-2-yl)-3-(piperidin-1-ylsulfonyl)benzamide

HRID 1967515Notes

Reaction equation

HRID 1967515 reaction equation
[N:1]1([S:7]([C:10]2[CH:11]=[C:12]([CH:16]=[CH:17][CH:18]=2)[C:13]([OH:15])=O)(=[O:9])=[O:8])[CH2:6][CH2:5][CH2:4][CH2:3][CH2:2]1.[CH3:19][O:20][C:21]1[C:22]([NH2:27])=[N:23][CH:24]=[CH:25][CH:26]=1>>[CH3:19][O:20][C:21]1[C:22]([NH:27][C:13](=[O:15])[C:12]2[CH:16]=[CH:17][CH:18]=[C:10]([S:7]([N:1]3[CH2:2][CH2:3][CH2:4][CH2:5][CH2:6]3)(=[O:8])=[O:9])[CH:11]=2)=[N:23][CH:24]=[CH:25][CH:26]=1

Participants

3

Reactant 2

HCID 7678893-(Piperidine-1-sulfonyl)benzoic acidHCID 99203842-Amino-3-methoxypyridine

Product 1

HCID 44468938N-(3-methoxypyridin-2-yl)-3-(piperidin-1-ylsulfonyl)benzamide

Procedure

The entitled compound was produced according to the method of Example 92 but using 3-(piperidin-1-ylsulfonyl)benzoic acid and 3-methoxypyridine-2-amine as the starting materials.

Workup

  1. customThe entitled compound was produced

Sources & evidence

ORD record
ord-94f3e1a3cbf34b978f39c3250fbf9f63
Source dataset
uspto-grants-2013_04
Patent number
US08420823B2

Reaction notes

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