3-(Piperidine-1-sulfonyl)benzoic acid → HCID 178510602, compound

HRID 1967528Notes

Reaction equation

HRID 1967528 reaction equation
[N:1]1([S:7]([C:10]2[CH:11]=[C:12]([CH:16]=[CH:17][CH:18]=2)[C:13]([OH:15])=O)(=[O:9])=[O:8])[CH2:6][CH2:5][CH2:4][CH2:3][CH2:2]1.[NH2:19][C:20]1[NH:24][CH:23]=[N:22][C:21]=1[C:25]#[N:26]>>[C:25]([C:21]1[N:22]=[CH:23][NH:24][C:20]=1[NH:19][C:13](=[O:15])[C:12]1[CH:16]=[CH:17][CH:18]=[C:10]([S:7]([N:1]2[CH2:2][CH2:3][CH2:4][CH2:5][CH2:6]2)(=[O:8])=[O:9])[CH:11]=1)#[N:26]

Participants

3

Reactant 2

HCID 7678893-(Piperidine-1-sulfonyl)benzoic acidHCID 178510601HCID 178510601, compound

Product 1

HCID 178510602HCID 178510602, compound

Procedure

The entitled compound was produced according to the method of Example 92 but using 3-(piperidin-1-ylsulfonyl)benzoic acid and 5-amino-1H-imidazole-4-carbonitrile as the starting materials.

Workup

  1. customThe entitled compound was produced

Sources & evidence

ORD record
ord-438febc0824b4ba285a878448addf289
Source dataset
uspto-grants-2013_04
Patent number
US08420823B2

Reaction notes

Loading…