3-(Pyrrolidine-1-sulfonyl)benzoic acid → HCID 178521742, compound

HRID 1967529Notes

Reaction equation

HRID 1967529 reaction equation
[N:1]1([S:6]([C:9]2[CH:10]=[C:11]([CH:15]=[CH:16][CH:17]=2)[C:12]([OH:14])=O)(=[O:8])=[O:7])[CH2:5][CH2:4][CH2:3][CH2:2]1.[CH:18]1([C:21]2[NH:25][N:24]=[C:23]([NH2:26])[CH:22]=2)[CH2:20][CH2:19]1>>[CH:18]1([C:21]2[CH:22]=[C:23]([NH:26][C:12](=[O:14])[C:11]3[CH:15]=[CH:16][CH:17]=[C:9]([S:6]([N:1]4[CH2:2][CH2:3][CH2:4][CH2:5]4)(=[O:7])=[O:8])[CH:10]=3)[NH:24][N:25]=2)[CH2:20][CH2:19]1

Participants

3

Reactant 2

HCID 7676903-(Pyrrolidine-1-sulfonyl)benzoic acidHCID 27580143-cyclopropyl-1H-pyrazol-5-amine

Product 1

HCID 178521742HCID 178521742, compound

Procedure

The entitled compound was produced according to the method of Example 92 but using 3-(pyrrolidin-1-ylsulfonyl)benzoic acid and 5-cyclopropyl-1H-pyrazole-3-amine as the starting materials.

Workup

  1. customThe entitled compound was produced

Sources & evidence

ORD record
ord-fc81df3c632c4bc98df52e7604758a1f
Source dataset
uspto-grants-2013_04
Patent number
US08420823B2

Reaction notes

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