2-Cyclopropyl-1-fluoro-4-iodobenzene → 3-Cyclopropyl-N-[[4-(1,1-dimethylethyl)phenyl]methyl]-4-fluorobenzeneethanamine

Beteiligte Stoffe

Reaktionsschritte

The title compound was synthesized in analogy to example S6-C using 2-cyclopropyl-1-fluoro-4-iodobenzene (100 mg, 0.38 mmol) and 3-(4-tert-butylbenzyl)-[1,2,3]oxathiazolidine 2,2-dioxide (103 mg, 0.38 mmol). The residue was purified by flash column chromatography to give the desired product (35 mg, 28%) as a colorless oil. MS (ISP) 326.3 (M+H)+.

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