HuagongsheHuagongshe Chemistry Print Report · For research reference only
Pyrazole → HCID 16722360, compound
Participants
| Role | Name | HCID | Charge |
|---|---|---|---|
| Reactant | Pyrazole | HCID 1048 | — |
| Reactant | HCID 16723117 | HCID 16723117 | — |
| Product | HCID 16722360 | HCID 16722360 | 79% |
Reaction Steps
As described for example 106, 4-{4-[5-(5-chloro-3-phenyl-isoxazol-4-yl)-[1,3,4]oxadiazol-2-yl]-3-methoxy-phenyl}-morpholine (100 mg, 0.23 mmol) using pyrazole instead of dimethylamine hydrochloride was converted to the title compound (85 mg, 79%) which was obtained as an off-white solid. MS: m/e=471.3 [M+H]+.
Provenance & Evidence
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| Patent number | US07541372B2 |
| Source dataset | uspto-grants-2009_06 |
| ORD ID | ord-bfc6984a571d46e5bddc7026b4ae05c3 |
| Source note | uspto-grants-2009_06 |