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HuagongsheHuagongshe Chemistry Print Report · For research reference only
HRID 1984805Generated: November 4, 2026

3-Chloro-4-fluorophenylboronic Acid (contains varying amounts of Anhydride) → HCID 10480005, compound

https://huagongshe.com/reaction/1984805

Reaction equation

Participants

RoleNameHCIDCharge
Reactant3-Chloro-4-fluorophenylboronic Acid (contains varying amounts of Anhydride)HCID 2734660—
ReactantHCID 58717891HCID 58717891—
ProductHCID 10480005HCID 1048000581.6%

Reaction Steps

3-Biphenyl-4-yl-(2S)-[(5-bromo-benzoyl-amino)-propionic acid (100 mg, 0.23 mmol) was reacted with 3-chloro-4-fluoro-phenyl boronic acid (0.123 mg, 0.69 mmol) by following general procedure D to afford title compound (89 mg) as a white solid.

Provenance & Evidence

DOI10.6084/m9.figshare.5104873.v1
Patent numberUS07544699B2
Source datasetuspto-grants-2009_06
ORD IDord-780ea1a677ae4d248d9d4adef7813cfa
Source noteuspto-grants-2009_06