5-Azaindole → HCID 66922198, compound

HRID 2039821Notes

Reaction equation

[NH:1]1[C:9]2[C:4](=[CH:5][N:6]=[CH:7][CH:8]=2)[CH:3]=[CH:2]1.[F:10][C:11]1[CH:16]=[CH:15][C:14](I)=[CH:13][CH:12]=1>>[F:10][C:11]1[CH:16]=[CH:15][C:14]([N:1]2[C:9]3[CH:8]=[CH:7][N:6]=[CH:5][C:4]=3[CH:3]=[CH:2]2)=[CH:13][CH:12]=1

Participants

Reactant 2

HCID 92205-Azaindole

HCID 96054-Fluoroiodobenzene

Product 1

HCID 66922198HCID 66922198, compound

Procedure

The title compound was prepared from 5-azaindole (1.00 g, 8.47 mmol) and 1-fluoro-4-iodobenzene analogously as described in example 1, step 1. Yield: 1.23 g.

Sources & evidence

ORD record: ord-262fde32cc4f46568e3af575544c337e
Source dataset: uspto-grants-2013_11
DOI: 10.6084/m9.figshare.5104873.v1
Patent number: US08580813B2

Reaction notes

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