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HuagongsheHuagongshe Chemistry Print Report · For research reference only
HRID 2046502Generated: October 26, 2026

3-Pyridinylboronic acid → 2-Amino-4-methyl-7-(2-pyridin-3-yl-phenyl)-7,8-dihydro-6H-quinazolin-5-one

https://huagongshe.com/reaction/2046502

Reaction equation

Participants

RoleNameHCIDCharge
Reactant3-Pyridinylboronic acidHCID 2734378—
Reactant2-amino-7-biphenyl-2-yl-4-methyl-7,8-dihydro-6H-quinazolin-5-oneHCID 58269344—
ReactantHCID 178430661HCID 178430661—
Product2-Amino-4-methyl-7-(2-pyridin-3-yl-phenyl)-7,8-dihydro-6H-quinazolin-5-oneHCID 58269357—

Reaction Steps

The title compound was prepared from 2-amino-4-methyl-7-(2-bromo-phenyl)-4-methyl-7,8-dihydro-6H-quinazolin-5-one (example 3/i stage 2/3) and pyridin-3-ylboronic acid, following the procedure describing the synthesis of 2-amino-7-biphenyl-2-yl-4-methyl-7,8-dihydro-6H-quinazolin-5-one (example 5/a stage 1).

Provenance & Evidence

DOI10.6084/m9.figshare.5104873.v1
Patent numberUS08592430B2
Source datasetuspto-grants-2013_11
ORD IDord-9fa461ccdf6b43c1998aeec23a2f9fd1
Source noteuspto-grants-2013_11