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HuagongsheHuagongshe Chemistry Print Report · For research reference only
HRID 2061128Generated: November 2, 2026

3-Methoxybenzenethiol → 3-(2-Fluoro-3-aminobenzyl)-7-methyloxy-4-methyl-2-oxo-2H-1-benzothiopyran

https://huagongshe.com/reaction/2061128

Reaction equation

Participants

RoleNameHCIDCharge
Reactant3-MethoxybenzenethiolHCID 84989—
Reactant2-(2-Fluoro-3-aminobenzyl)-3-oxobutanoic acid ethyl esterHCID 66860353—
Product3-(2-Fluoro-3-aminobenzyl)-7-methyloxy-4-methyl-2-oxo-2H-1-benzothiopyranHCID 58232224—

Reaction Steps

The title compound was synthesized using 3-methyloxy-benzenethiol and 2-(2-fluoro-3-aminobenzyl)-3-oxobutanoic acid ethyl ester under the same conditions as in the manufacturing example for compound 5d-0-4S1.

Provenance & Evidence

DOI10.6084/m9.figshare.5104873.v1
Patent numberUS08278465B2
Source datasetuspto-grants-2012_10
ORD IDord-3617c94cb92c4bfea4961303eb16d915
Source noteuspto-grants-2012_10