1-[5-(2-Methyl-[1,3]dioxolan-2-yl)-furan-2-ylmethyl]-1H-pyrazol-3-ylamine → HCID 66928174, compound

HRID 2065357Notes

Reaction equation

HRID 2065357 reaction equation
[CH3:1][C:2]1([C:7]2[O:11][C:10]([CH2:12][N:13]3[CH:17]=[CH:16][C:15]([NH2:18])=[N:14]3)=[CH:9][CH:8]=2)[O:6]CCO1.[CH:19]([O:22][CH2:23][CH2:24][C:25]1[CH:26]=[C:27]([C:31]2[O:35][CH:34]=[N:33][C:32]=2[C:36](O)=[O:37])[CH:28]=[CH:29][CH:30]=1)([CH3:21])[CH3:20]>>[C:2]([C:7]1[O:11][C:10]([CH2:12][N:13]2[CH:17]=[CH:16][C:15]([NH:18][C:36]([C:32]3[N:33]=[CH:34][O:35][C:31]=3[C:27]3[CH:28]=[CH:29][CH:30]=[C:25]([CH2:24][CH2:23][O:22][CH:19]([CH3:21])[CH3:20])[CH:26]=3)=[O:37])=[N:14]2)=[CH:9][CH:8]=1)(=[O:6])[CH3:1]

Participants

3

Procedure

Following general procedure B followed by C, starting from 1-[5-(2-methyl-[1,3]dioxolan-2-yl)-furan-2-ylmethyl]-1H-pyrazol-3-ylamine and 5-[3-(2-isopropoxy-ethyl)-phenyl]-oxazole-4-carboxylic acid. LC-MS-conditions 02: tR=1.04 min; [M+H]+=463.35.

Sources & evidence

ORD record
ord-02677422cb6149ab89d1cffdb291e765
Source dataset
uspto-grants-2012_10
Patent number
US08288419B2

Reaction notes

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