Benzocaine → HCID 16776736, compound

HRID 2073752Notes

Reaction equation

HRID 2073752 reaction equation
[NH2:1][C:2]1[CH:12]=[CH:11][C:5]([C:6]([O:8]CC)=[O:7])=[CH:4][CH:3]=1.[CH2:13]([S:17](Cl)(=[O:19])=[O:18])[CH2:14][CH2:15][CH3:16]>N1C=CC=CC=1>[CH2:13]([S:17]([NH:1][C:2]1[CH:3]=[CH:4][C:5]([C:6]([OH:8])=[O:7])=[CH:11][CH:12]=1)(=[O:19])=[O:18])[CH2:14][CH2:15][CH3:16]

Participants

4

Reactant 2

HCID 2337BenzocaineHCID 754301-Butanesulfonyl chloride

Product 1

HCID 16776736HCID 16776736, compound

Reagents, catalysts & solvents 1

HCID 1049PyridineSolvent

Procedure

In a manner similar to Preparation 9 react ethyl 4-aminobenzoate with 1-butanesulfonyl chloride and pyridine to obtain the title compound.

Workup

  1. customIn a manner similar to Preparation 9

Sources & evidence

ORD record
ord-ce210b3cf42544aebf66091f12c7495b
Source dataset
uspto-grants-1990_04
Patent number
US04920116

Reaction notes

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