Ethyl 3-{[(4-aminophenyl)carbonyl](methyl)amino}propanoate → 3-[({4-[(cyclohexyl{3-propyl-1-[5-(trifluoromethyl)pyridin-2-yl]-1H-pyrazol-4-yl}methyl)amino]phenyl}carbonyl)(methyl)amino]propanoic acid

Participants

Reaction Steps

Using cyclohexyl{3-propyl-1-[5-(trifluoromethyl)pyridin-2-yl]-1H-pyrazol-4-yl}methanol (0.65 g) synthesized in Example 5(3) and ethyl 3-{[(4-aminophenyl)carbonyl](methyl)amino}propanoate (0.44 g) synthesized in Example 2(2) and in the same manner as in Example 1(7), the title object compound (0.34 g, 34%) was obtained as a white solid.

Provenance & Evidence