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HuagongsheHuagongshe Chemistry Print Report · For research reference only
HRID 2093408Generated: November 1, 2026

4-(4,4,5,5-Tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-indazole → HCID 44543766, compound

https://huagongshe.com/reaction/2093408

Reaction equation

Participants

RoleNameHCIDCharge
Reactant4-(4,4,5,5-Tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-indazoleHCID 45480186—
Reactant2-Chloro-9-methyl-6-(4-morpholinyl)-9H-purineHCID 71500687—
ProductHCID 44543766HCID 44543766—

Reaction Steps

4-(2-Chloro-9-methyl-9H-purin-6-yl)morpholine (20 mg) was reacted with 4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-indazole via General Procedure A and purified via reverse phase HPLC to give 13.8 mg of 129 as a white solid. MS (Q1) 336.2 (M)+

Provenance & Evidence

DOI10.6084/m9.figshare.5104873.v1
Patent numberUS08445487B2
Source datasetuspto-grants-2013_05
ORD IDord-b811444487074a4da3853508e185fcc5
Source noteuspto-grants-2013_05