HCID 58154279, compound → HCID 44476132, compound

Participants

Reaction Steps

Obtained as a white solid (16%, exact isomeric form not determined) from 7-iodo-6-methyl-1,2-benzisoxazol-3-amine (preparation 24) and 4-(2-morpholinoethoxy)-6′-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)spiro[cyclohexane-1,3′-indolin]-2′-one (preparation 15) following the experimental procedure as described in example 1 followed by purification by flash chromatography (97:3 dichloromethane/methanol).

Provenance & Evidence