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HuagongsheHuagongshe Chemistry Print Report · For research reference only
HRID 2098749Generated: October 29, 2026

5-Indolylboronic acid → HCID 59593093, compound

https://huagongshe.com/reaction/2098749

Reaction equation

Participants

RoleNameHCIDCharge
Reactant5-Indolylboronic acidHCID 2734361—
Reactant2-Chloro-4-(morpholin-4-yl)thieno(3,2-d)pyrimidineHCID 20284971—
ProductHCID 59593093HCID 59593093—

Reaction Steps

2-Chloro-4-moropholinothieno[3.2-d]pyrimidine 4 was reacted with 5-indole boronic acid in General Procedure A on a 23.5 mmol scale to give 25.7 mg. of 271 after RP-HPLC purification. MS (Q1) 337.1 (M)+.

Provenance & Evidence

DOI10.6084/m9.figshare.5104873.v1
Patent numberUS08450315B2
Source datasetuspto-grants-2013_05
ORD IDord-b5f09cc91192499b86a75cae2707b245
Source noteuspto-grants-2013_05