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HuagongsheHuagongshe Chemistry Print Report · For research reference only
HRID 2098884Generated: November 1, 2026

4-(4,4,5,5-Tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-indazole → HCID 24970248, compound

https://huagongshe.com/reaction/2098884

Reaction equation

Participants

RoleNameHCIDCharge
Reactant4-(4,4,5,5-Tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-indazoleHCID 45480186—
ReactantHCID 86618458HCID 86618458—
ProductHCID 24970248HCID 24970248—

Reaction Steps

1-(2-Chloro-4-morpholinothieno[3,2-d]pyrimidin-6-yl)pyrrolidin-2-one (35 mg) was coupled to 4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-indazole via Procedure A. The product was purified by reverse phase HPLC to yield 19.5 mg of 438. MS (Q1) 421 (M)+

Provenance & Evidence

DOI10.6084/m9.figshare.5104873.v1
Patent numberUS08450315B2
Source datasetuspto-grants-2013_05
ORD IDord-85af3553d65e4cd59c8a47d7683e90b8
Source noteuspto-grants-2013_05