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HuagongsheHuagongshe Chemistry Print Report · For research reference only
HRID 2106848Generated: October 26, 2026

N-Formylleucine → (R,R,S,S)-Orlistat

https://huagongshe.com/reaction/2106848

Reaction equation

Participants

RoleNameHCIDCharge
ReactantN-FormylleucineHCID 9880216—
Reactant(2R,3S,4S)-3-Hexyl-4-(2-hydroxy-hex-5-enyl)-oxetan-2-oneHCID 53798423—
Product(R,R,S,S)-OrlistatHCID 16760542—

Reaction Steps

by esterifying (S)-3-hexyl-(S)-4-[(R)-2-hydroxy-5-hexenyl)-2-oxetanone with N-formyl-L-leucine there was obtained

Provenance & Evidence

DOI10.6084/m9.figshare.5104873.v1
Patent numberUS04931463
Source datasetuspto-grants-1990_06
ORD IDord-d89be49a929d4769a92fab12a57a226a
Source noteuspto-grants-1990_06