4-Methyl-3-(4-pyridin-3-yl-1,2,3-triazol-1-yl)-benzoic acid → N-(5-tert-Butyl-3-{[(2-dimethylamino-ethyl)-methyl-amino]-methyl}-2-methoxy-phenyl)-4-methyl-3-(4-pyridin-3-yl-[1,2,3]triazol-1-yl)-benzamide

Beteiligte Stoffe

Rolle	Name	HCID	Einwaage
Edukt	4-Methyl-3-(4-pyridin-3-yl-1,2,3-triazol-1-yl)-benzoic acid	HCID 21097331	—
Edukt	N-(3-amino-5-tert-butyl-2-methoxy-benzyl)-N,N',N'-trimethyl-ethane-1,2-diamine	HCID 21097366	—
Produkt	N-(5-tert-Butyl-3-{[(2-dimethylamino-ethyl)-methyl-amino]-methyl}-2-methoxy-phenyl)-4-methyl-3-(4-pyridin-3-yl-[1,2,3]triazol-1-yl)-benzamide	HCID 21097109	—

Reaktionsschritte

Example 10 was prepared by coupling 4-methyl-3-(4-pyridin-3-yl-[1,2,3]triazol-1-yl)-benzoic acid with N-(3-amino-5-tert-butyl-2-methoxy-benzyl)-N,N′,N′-trimethyl-ethane-1,2-diamine (see U.S. provisional application 60/526,569) in the same manner as Example 1. ESI MS m/z 554 [C32H41N7O2—H]−.

Herkunft & Nachweise

DOI	10.6084/m9.figshare.5104873.v1
Patentnummer	US07514458B2
Quelldatensatz	uspto-grants-2009_04
ORD ID	ord-161a494dfc36452284c6067b6bb6d521
Quellennotiz	uspto-grants-2009_04