Back
HuagongsheHuagongshe Chemistry Print Report · For research reference only
HRID 2109213Generated: October 25, 2026

3-Azido-4-methylbenzoic acid → 3-Azido-N-[3-methanesulfonylamino-2-methoxy-5-(1-methyl-cyclopropyl)-phenyl]-4-methyl-benzamide

https://huagongshe.com/reaction/2109213

Reaction equation

Participants

RoleNameHCIDCharge
Reactant3-Azido-4-methylbenzoic acidHCID 17973091—
Reactant3-azido-N-(5-tert-butyl-3-methanesulfonylamino-2-methoxy-phenyl)-4-methyl-benzamideHCID 21079202—
ReactantN-[3-amino-2-methoxy-5-(1-methyl-cyclopropyl)-phenyl]-methanesulfonamideHCID 22025264—
Product3-Azido-N-[3-methanesulfonylamino-2-methoxy-5-(1-methyl-cyclopropyl)-phenyl]-4-methyl-benzamideHCID 21097299—

Reaction Steps

3-Azido-N-[3-methanesulfonylamino-2-methoxy-5-(1-methyl-cyclopropyl)-phenyl]-4-methyl-benzamide was prepared from 3-azido-4-methyl benzoic acid and N-[3-amino-2-methoxy-5-(1-methyl-cyclopropyl)-phenyl]-methanesulfonamide in the same manner as 3-azido-N-(5-tert-butyl-3-methanesulfonylamino-2-methoxy-phenyl)-4-methyl-benzamide (Example 15).

Provenance & Evidence

DOI10.6084/m9.figshare.5104873.v1
Patent numberUS07514458B2
Source datasetuspto-grants-2009_04
ORD IDord-2ff27d46a4b540f5bbf7f5783e48d4c4
Source noteuspto-grants-2009_04