HCID 9997955, compound → HCID 11559626, compound

HRID 2112285Notes

Reaction equation

HRID 2112285 reaction equation
[C:1]1([C:7]2[N:8]=[C:9]([CH2:18][CH2:19][CH2:20][CH2:21][CH2:22][CH2:23][C:24]([OH:26])=O)[O:10][C:11]=2[C:12]2[CH:17]=[CH:16][CH:15]=[CH:14][CH:13]=2)[CH:6]=[CH:5][CH:4]=[CH:3][CH:2]=1.CC(C1C=CC(C2OC(CCCCCC([NH:49][OH:50])=O)=NC=2C2C=CC=CC=2)=CC=1)(C)C>>[OH:50][NH:49][C:24](=[O:26])[CH2:23][CH2:22][CH2:21][CH2:20][CH2:19][CH2:18][C:9]1[O:10][C:11]([C:12]2[CH:17]=[CH:16][CH:15]=[CH:14][CH:13]=2)=[C:7]([C:1]2[CH:6]=[CH:5][CH:4]=[CH:3][CH:2]=2)[N:8]=1

Participants

3

Reactant 2

HCID 9997955HCID 9997955, compoundHCID 11502359HCID 11502359, compound

Product 1

HCID 11559626HCID 11559626, compound

Procedure

Using 4,5-diphenyl-2-oxazoleheptanoic acid (653 mg), a reaction and a treatment were carried out in the same manner as in the section (3) of example 1 to obtain the desired subject compound 24 (530 mg, Y=77.8%).

Workup

  1. customa reaction
  2. customto obtain the

Sources & evidence

ORD record
ord-31318e7074c64f969b38a0585dc602eb
Source dataset
uspto-grants-2009_04
Patent number
US07521563B2

Reaction notes

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