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HuagongsheHuagongshe Chemistry Print Report · For research reference only
HRID 2113002Generated: October 27, 2026

(2H-1,3-benzodioxol-5-yl)boronic acid → 3-(4-Benzo[1,3]dioxol-5-yl-phenoxymethyl)-benzoic acid

https://huagongshe.com/reaction/2113002

Reaction equation

Participants

RoleNameHCIDCharge
Reactant(2H-1,3-benzodioxol-5-yl)boronic acidHCID 2734371—
ReactantMethyl 3-((4-iodophenoxy)methyl)benzoateHCID 57643351—
Product3-(4-Benzo[1,3]dioxol-5-yl-phenoxymethyl)-benzoic acidHCID 11645963—

Reaction Steps

3-(4-Benzo[1,3]dioxol-5-yl-phenoxymethyl)-benzoic acid was prepared using general procedure 1 from 3-(4-iodo-phenoxymethyl)-benzoic acid methyl ester (of Intermediate 1) and 3,4-methylenedioxybenzeneboronic acid (ASDI Incorporated, Newark, Del.). Mass spectrum MH+=349.

Provenance & Evidence

DOI10.6084/m9.figshare.5104873.v1
Patent numberUS07524870B2
Source datasetuspto-grants-2009_04
ORD IDord-c83b632a975a4d689bddfbbb5b826a39
Source noteuspto-grants-2009_04