3-Benzylsulfonylamino-6-methyl-1-carboxymethyl-2-pyridinone → HCID 44337785, compound

HRID 2113048Notes

Reaction equation

HRID 2113048 reaction equation
[CH2:1]([S:8]([NH:11][C:12]1[C:13](=[O:23])[N:14]([CH2:19][C:20]([OH:22])=O)[C:15]([CH3:18])=[CH:16][CH:17]=1)(=[O:10])=[O:9])[C:2]1[CH:7]=[CH:6][CH:5]=[CH:4][CH:3]=1.Cl.[CH3:25][N:26]1[CH:34]=[C:33]2[C:28]([CH2:29][CH2:30][CH:31]([CH2:35][NH2:36])[CH2:32]2)=[N:27]1>>[CH2:1]([S:8]([NH:11][C:12]1[C:13](=[O:23])[N:14]([CH2:19][C:20]([NH:36][CH2:35][CH:31]2[CH2:30][CH2:29][C:28]3[C:33](=[CH:34][N:26]([CH3:25])[N:27]=3)[CH2:32]2)=[O:22])[C:15]([CH3:18])=[CH:16][CH:17]=1)(=[O:10])=[O:9])[C:2]1[CH:3]=[CH:4][CH:5]=[CH:6][CH:7]=1

Participants

3

Reactant 2

HCID 154582213-Benzylsulfonylamino-6-methyl-1-carboxymethyl-2-pyridinoneHCID 690368382-methyl-4,5,6,7-tetrahydro-2H-indazol-5-ylmethanamine hydrochloride

Product 1

HCID 44337785HCID 44337785, compound

Procedure

The title compound was prepared from 2-[3-[(benzylsulfonyl)amino]-6 -methyl-2-oxo-1(2H)-pyridinyl]acetic acid and 2-methyl-4,5,6,7-tetrahydro-2H-indazol-5-ylmethanamine hydrochloride using the procedure of EXAMPLE 1 (STEP 6), and was obtained as a faint yellow solid compound.

Workup

  1. customwas obtained as a faint yellow solid compound

Sources & evidence

ORD record
ord-685b0a5e116842a9925ca73ce22c6015
Source dataset
uspto-grants-2009_04
Patent number
US07524871B2

Reaction notes

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