4-Aminocarbonylphenylboronic acid → HCID 46846504, compound

Participants

Reaction Steps

4′-[(1R)-1-[[(6,7-dichloro-3-oxo-2,3-dihydro-4H-1,4-benzoxazin-4-yl)acetyl](methyl)amino]-2-(1-pyrrolidinyl)ethyl]-4-biphenylcarboxamide was prepared in a similar manner as in the preparation of 4′-[(1R)-1-[[(6,7-dichloro-3-oxo-2,3-dihydro-4H-1,4-benzoxazin-4-yl)acetyl](methyl)amino]-2-(1-pyrrolidinyl)ethyl]-3-biphenylcarboxamide except replacing [3-(aminocarbonyl)phenyl]boronic acid with [4-(aminocarbonyl)phenyl]boronic acid. As is appreciated by those skilled in the art, this analogous example may involve variations in synthetic procedure.

Provenance & Evidence