5-Amino-2,3-dihydro-1,3-benzoxazol-2-one → HCID 69100683, compound

HRID 2115148Notes

Reaction equation

HRID 2115148 reaction equation
[NH2:1][C:2]1[CH:3]=[CH:4][C:5]2[O:9][C:8](=[O:10])[NH:7][C:6]=2[CH:11]=1.[CH2:12]([CH:19]1[CH2:24][CH2:23][N:22]([C:25](=[O:29])[C:26](O)=[O:27])[CH2:21][CH2:20]1)[C:13]1[CH:18]=[CH:17][CH:16]=[CH:15][CH:14]=1>O>[CH2:12]([CH:19]1[CH2:20][CH2:21][N:22]([C:25](=[O:29])[C:26]([NH:1][C:2]2[CH:3]=[CH:4][C:5]3[O:9][C:8](=[O:10])[NH:7][C:6]=3[CH:11]=2)=[O:27])[CH2:23][CH2:24]1)[C:13]1[CH:14]=[CH:15][CH:16]=[CH:17][CH:18]=1

Participants

4

Reactant 2

HCID 268565-Amino-2,3-dihydro-1,3-benzoxazol-2-oneHCID 16110264(4-Benzylpiperidin-1-yl)oxoacetic acid

Product 1

HCID 69100683HCID 69100683, compound

Reagents, catalysts & solvents 1

HCID 962WaterSolvent

Procedure

The title compound is prepared from 5-amino-3H-benzoxazole-2-one and (4-benzyl-piperidin-1-yl)-oxo-acetic acid (Example 5b) according to the method described in Example 2. Melting Point: 187-190° C. (water)

Sources & evidence

ORD record
ord-c1de862d1c95479b94eec769e5d19840
Source dataset
uspto-grants-2008_10
Patent number
US07435744B2

Reaction notes

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