HCID 23442400, compound → HCID 10267948, compound

HRID 2119632Notes

Reaction equation

HRID 2119632 reaction equation
[NH2:1][C:2]1[CH:7]=[CH:6][C:5]([CH2:8][C:9]2[CH:14]=[CH:13][C:12]([O:15][CH3:16])=[CH:11][CH:10]=2)=[CH:4][C:3]=1[C:17]([C:19]1[N:23]([CH3:24])[N:22]=[CH:21][C:20]=1I)=[O:18].NC1C=CC(CC2C=CC(Cl)=CC=2)=CC=1C(C1N(C)N=CC=1I)=O>>[CH3:16][O:15][C:12]1[CH:13]=[CH:14][C:9]([CH2:8][C:5]2[CH:6]=[CH:7][C:2]3[NH:1][C:20]4[CH:21]=[N:22][N:23]([CH3:24])[C:19]=4[C:17](=[O:18])[C:3]=3[CH:4]=2)=[CH:10][CH:11]=1

Participants

3

Reactant 2

HCID 23442400HCID 23442400, compoundHCID 23442449HCID 23442449, compound

Product 1

HCID 10267948HCID 10267948, compound

Procedure

The title compound was prepared according to the procedure of step 6 in EXAMPLE 13 using [2-amino-5-(4-methoxybenzyl)phenyl](4-iodo-1-methyl-1H-pyrazol-5-yl)methanone (EXAMPLE 16, step 4), instead of [2-amino-5-(4-chlorobenzyl)phenyl](4-iodo-1-methyl-1H-pyrazol-5-yl)methanone.

Sources & evidence

ORD record
ord-5f558591947f49a78e46b0d479c29e33
Source dataset
uspto-grants-2004_02
Patent number
US06686373B2

Reaction notes

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