HCID 23442310, compound → HCID 23442342, compound

HRID 2119637Notes

Reaction equation

HRID 2119637 reaction equation
[NH2:1][C:2]1[CH:7]=[CH:6][C:5]([CH2:8][C:9]2[CH:14]=[CH:13][CH:12]=[CH:11][C:10]=2[O:15][CH3:16])=[CH:4][C:3]=1[C:17]([C:19]1[N:23]([CH3:24])[N:22]=[CH:21][C:20]=1I)=[O:18].NC1C=CC(CC2C=CC(Cl)=CC=2)=CC=1C(C1N(C)N=CC=1I)=O>>[CH3:16][O:15][C:10]1[CH:11]=[CH:12][CH:13]=[CH:14][C:9]=1[CH2:8][C:5]1[CH:6]=[CH:7][C:2]2[NH:1][C:20]3[CH:21]=[N:22][N:23]([CH3:24])[C:19]=3[C:17](=[O:18])[C:3]=2[CH:4]=1

Participants

3

Reactant 2

HCID 23442310HCID 23442310, compoundHCID 23442449HCID 23442449, compound

Product 1

HCID 23442342HCID 23442342, compound

Procedure

The title compound was prepared according to the procedure of step 6 in EXAMPLE 13 using [2-amino-5-(2-methoxybenzyl)phenyl](4-iodo-1-methyl-1H-pyrazol-5-yl)methanone (EXAMPLE 21, step 4), instead of [2-amino-5-(4-chlorobenzyl)phenyl](4-iodo-1-methyl-1H-pyrazol-5-yl)methanone.

Sources & evidence

ORD record
ord-cb03e49f591546a982ea8394c4b3b08b
Source dataset
uspto-grants-2004_02
Patent number
US06686373B2

Reaction notes

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