HCID 71075457, compound → HCID 71099832, compound

HRID 2170722Notes

Reaction equation

HRID 2170722 reaction equation
[CH3:1][O:2][C:3]([C:5]1[CH:6]=[C:7]([CH:23]=[CH:24][CH:25]=1)[CH2:8][N:9]1[C:17]2[C:12](=[CH:13][C:14]([C:18]([OH:20])=O)=[CH:15][CH:16]=2)[C:11]([CH3:21])=[C:10]1[CH3:22])=[O:4].[CH:26]1([C:29]2[CH:30]=[C:31]([C@@H:35]([NH2:37])[CH3:36])[CH:32]=[CH:33][CH:34]=2)[CH2:28][CH2:27]1>>[CH:26]1([C:29]2[CH:30]=[C:31]([C@@H:35]([NH:37][C:18]([C:14]3[CH:13]=[C:12]4[C:17](=[CH:16][CH:15]=3)[N:9]([CH2:8][C:7]3[CH:6]=[C:5]([CH:25]=[CH:24][CH:23]=3)[C:3]([O:2][CH3:1])=[O:4])[C:10]([CH3:22])=[C:11]4[CH3:21])=[O:20])[CH3:36])[CH:32]=[CH:33][CH:34]=2)[CH2:28][CH2:27]1

Participants

3

Reactant 2

HCID 71075457HCID 71075457, compoundHCID 86674583(αS)-3-Cyclopropyl-α-methylbenzenemethanamine

Product 1

HCID 71099832HCID 71099832, compound

Procedure

The title compound was prepared following the same general protocol as described in Step 5, Example 35, using 1-(3-(methoxycarbonyl)benzyl)-2,3-dimethyl-1H-indole-5-carboxylic acid and (S)-1-(3-cyclopropylphenyl)ethanamine.

Sources & evidence

ORD record
ord-2fe841b5ac894da59d5617a2a80ae39c
Source dataset
uspto-grants-2015_06
Patent number
US09051265B2

Reaction notes

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