Methyl azetidine-3-carboxylate → 1-(Propane-1-sulfonyl)-azetidine-3-carboxylic acid methyl ester

HRID 2177124Notes

Reaction equation

HRID 2177124 reaction equation
[CH3:1][O:2][C:3]([CH:5]1[CH2:8][NH:7][CH2:6]1)=[O:4].C1(N[S:13]([CH2:16][CH2:17][CH3:18])(=[O:15])=[O:14])CC1>>[CH3:1][O:2][C:3]([CH:5]1[CH2:8][N:7]([S:13]([CH2:16][CH2:17][CH3:18])(=[O:15])=[O:14])[CH2:6]1)=[O:4]

Participants

3

Reactant 2

HCID 20132751Methyl azetidine-3-carboxylateHCID 59547736Propane-1-Sulfonic Acid Cyclopropyl Amide

Product 1

HCID 574714481-(Propane-1-sulfonyl)-azetidine-3-carboxylic acid methyl ester

Procedure

Prepared by standard procedure from azetidine-3-carboxylic acid methyl ester and propane-1-sulfonyl chloride (e.g. example 279).

Sources & evidence

ORD record
ord-cdf365e963604fe686e270fcc3aeb50b
Source dataset
uspto-grants-2015_06
Patent number
US09067871B2

Reaction notes

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