HCID 86271308, compound → HCID 90409273, compound

HRID 2177645Notes

Reaction equation

HRID 2177645 reaction equation
[Cl:1][C:2]1[C:7]([C:8]([F:11])([F:10])[F:9])=[CH:6][CH:5]=[CH:4][C:3]=1[C:12]([N:14]1[CH:19]=[CH:18][C:17]2[N:20]([C:23]3[N:28]=[C:27]([CH3:29])[CH:26]=[CH:25][N:24]=3)[N:21]=[N:22][C:16]=2[CH:15]1[CH3:30])=[O:13].ClC1C(C(F)(F)F)=CC=CC=1C(N1C=CC2N(C3C=NC=CN=3)N=NC=2C1C)=O>>[Cl:1][C:2]1[C:7]([C:8]([F:9])([F:11])[F:10])=[CH:6][CH:5]=[CH:4][C:3]=1[C:12]([N:14]1[CH2:19][CH2:18][C:17]2[N:20]([C:23]3[N:28]=[C:27]([CH3:29])[CH:26]=[CH:25][N:24]=3)[N:21]=[N:22][C:16]=2[CH:15]1[CH3:30])=[O:13]

Participants

3

Reactant 2

HCID 86271308HCID 86271308, compoundHCID 90410971HCID 90410971, compound

Product 1

HCID 90409273HCID 90409273, compound

Procedure

The title compound was prepared in a manner analogous to Example 73 substituting the product of Example 252, Step 2 for the 5-{[2-chloro-3-(trifluoromethyl)phenyl]carbonyl}-4-methyl-1-pyrazin-2-yl-4,5-dihydro-1H-[1,2,3]triazolo[4,5-c]pyridine. MS (E S I) mass calcd. C19H16ClF3N6O, 436.1. m/z found, 437.1 [M+H]+.

Sources & evidence

ORD record
ord-6b483f62e48540d2bf41cf4b4eeaa18d
Source dataset
uspto-grants-2015_06
Patent number
US09066946B2

Reaction notes

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