Back
HuagongsheHuagongshe Chemistry Print Report · For research reference only
HRID 2177776Generated: October 30, 2026

Thiophene-3-boronic acid → Methyl 6-(benzenesulphonylmethyl)-2-methoxy-3-(thien-3-yl)benzoate

https://huagongshe.com/reaction/2177776

Reaction equation

Participants

RoleNameHCIDCharge
ReactantThiophene-3-boronic acidHCID 581760—
ReactantMethyl 6-(benzenesulfonylmethyl)-3-bromo-2-methoxybenzoateHCID 66685730—
ReactantEthyl 3-(furan-3-yl)-2-methoxy-6-(2-methylbenzenesulphonylmethyl)benzoateHCID 67107552—
ProductMethyl 6-(benzenesulphonylmethyl)-2-methoxy-3-(thien-3-yl)benzoateHCID 67107684—

Reaction Steps

Prepared by proceeding in a similar manner to Intermediate 28, starting from methyl 6-(benzenesulphonylmethyl)-3-bromo-2-methoxybenzoate (Intermediate 65) and thiophene-3-boronic acid.

Provenance & Evidence

DOI10.6084/m9.figshare.5104873.v1
Patent numberUS09067905B2
Source datasetuspto-grants-2015_06
ORD IDord-6385f31c88654115b8a2cf17e9f3f0fb
Source noteuspto-grants-2015_06