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HuagongsheHuagongshe Chemistry Print Report · For research reference only
HRID 2177841Generated: October 31, 2026

Furan-3-boronic acid → (Z)-methyl 6-((2-(3-(diethylamino)prop-1-enyl)-4-fluorobenzenesulfonyl)methyl)-3-(furan-3-yl)-2-hydroxybenzoate

https://huagongshe.com/reaction/2177841

Reaction equation

Participants

RoleNameHCIDCharge
ReactantFuran-3-boronic acidHCID 2734358—
Reactant(Z)-methyl 3-bromo-6-((2-(3-(diethylamino)prop-1-enyl)-4-fluorobenzenesulfonyl)methyl)-2-hydroxybenzoateHCID 66693503—
Reactant(Z)-methyl 6-((2-(3-(diethylamino)prop-1-enyl)-4-fluorobenzenesulfonyl)methyl)-3-(furan-3-yl)-2-methoxybenzoateHCID 69915014—
Product(Z)-methyl 6-((2-(3-(diethylamino)prop-1-enyl)-4-fluorobenzenesulfonyl)methyl)-3-(furan-3-yl)-2-hydroxybenzoateHCID 86677120—

Reaction Steps

Prepared by proceeding in a similar manner to Intermediate 160, starting from (Z)-methyl 3-bromo-6-((2-(3-(diethylamino)prop-1-enyl)-4-fluorobenzenesulfonyl)methyl)-2-hydroxybenzoate (Intermediate 197) and furan-3-boronic acid.

Provenance & Evidence

DOI10.6084/m9.figshare.5104873.v1
Patent numberUS09067905B2
Source datasetuspto-grants-2015_06
ORD IDord-dc9cbbdf33274665a329441a29bb17b4
Source noteuspto-grants-2015_06