6-(furan-3-yl)-5-methoxy-2-oxo-2-phenyl-1H-2-lambda*6*-benzo[d][1,2]thiazin-4-one → t-Butyl 3-(furan-3-yl)-2-methoxy-6-[(S-phenylsulphonimidoyl)methyl]benzoate

HRID 2177859Notes

Reaction equation

HRID 2177859 reaction equation
O1C=CC(C2C=CC3CS(=O)(C4C=CC=CC=4)=NC(=O)C=3C=2OC)=C1.[O:26]1[CH:30]=[CH:29][C:28]([C:31]2[C:32]([O:60][CH3:61])=[C:33]([C:41]([CH2:44][S:45]([C:54]3[CH:59]=[CH:58][CH:57]=[CH:56][CH:55]=3)(=[N:47]C(=O)C(F)(F)F)=[O:46])=[CH:42][CH:43]=2)[C:34]([O:36][C:37]([CH3:40])([CH3:39])[CH3:38])=[O:35])=[CH:27]1>>[O:26]1[CH:30]=[CH:29][C:28]([C:31]2[C:32]([O:60][CH3:61])=[C:33]([C:41]([CH2:44][S:45]([C:54]3[CH:59]=[CH:58][CH:57]=[CH:56][CH:55]=3)(=[NH:47])=[O:46])=[CH:42][CH:43]=2)[C:34]([O:36][C:37]([CH3:40])([CH3:39])[CH3:38])=[O:35])=[CH:27]1

Participants

3

Reactant 2

HCID 699150306-(furan-3-yl)-5-methoxy-2-oxo-2-phenyl-1H-2-lambda*6*-benzo[d][1,2]thiazin-4-oneHCID 86677128t-butyl 3-(furan-3-yl)-2-methoxy-6-{[S-phenyl-N-(trifluoroacetyl)sulphonimidoyl]methyl}benzoate2×

Product 1

HCID 86677127t-Butyl 3-(furan-3-yl)-2-methoxy-6-[(S-phenylsulphonimidoyl)methyl]benzoate

Procedure

Prepared by proceeding in a similar manner to Intermediate 214, starting from t-butyl 3-(furan-3-yl)-2-methoxy-6-{[S-phenyl-N-(trifluoroacetyl)sulphonimidoyl]methyl}benzoate (Intermediate 220).

Workup

  1. customPrepared

Sources & evidence

ORD record
ord-96a77afeae5a44d89a6c51ba30bb8ff8
Source dataset
uspto-grants-2015_06
Patent number
US09067905B2

Reaction notes

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