Tert-butyl 4-(2-methoxy-2-oxoethylidene)piperidine-1-carboxylate → HCID 59382660, compound

HRID 217961Notes

Reaction equation

HRID 217961 reaction equation
[CH3:1][O:2][CH2:3][CH2:4][N:5]1[CH2:10][CH2:9][C:8](=[CH:11][C:12]([O:14]C)=[O:13])[CH2:7][CH2:6]1.COC(C=C1CCN(C(OC(C)(C)C)=O)CC1)=O>>[CH3:1][O:2][CH2:3][CH2:4][N:5]1[CH2:6][CH2:7][C:8](=[CH:11][C:12]([OH:14])=[O:13])[CH2:9][CH2:10]1

Participants

3

Reactant 2

HCID 10377658Tert-butyl 4-(2-methoxy-2-oxoethylidene)piperidine-1-carboxylateHCID 59382747HCID 59382747, compound

Product 1

HCID 59382660HCID 59382660, compound

Procedure

The title compound was prepared following the procedure for the preparation of intermediate 3a except that methyl 2-(1-(2-methoxyethyl)piperidin-4-ylidene)acetate was substituted for tert-butyl 4-((methoxycarbonyl)methylene)piperidine-1-carboxylate.

Sources & evidence

ORD record
ord-ff8de619d87546a4bd7f05638e7b1fb4
Source dataset
uspto-grants-2012_06
Patent number
US08198301B2

Reaction notes

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