Boronic Acid → HCID 178440403, compound

HRID 2197406Notes

Reaction equation

HRID 2197406 reaction equation
Br[C:2]1[CH:10]=[CH:9][CH:8]=[C:7]2[C:3]=1[C:4]([CH:11]([CH3:13])[CH3:12])=[N:5][NH:6]2.[BH:14]([OH:16])[OH:15]>>[CH:11]([C:4]1[C:3]2[C:2]([B:14]([OH:16])[OH:15])=[CH:10][CH:9]=[CH:8][C:7]=2[NH:6][N:5]=1)([CH3:13])[CH3:12]

Participants

3

Reactant 2

HCID 61668Boronic AcidHCID 1784404044-Bromo-3-isopropyl-1H-indazole

Product 1

HCID 178440403HCID 178440403, compound

Procedure

4-Bromo-3-isopropyl-1H-indazole is converted to the corresponding boronic acid following analogous procedures to that given in the preceding example. 1H NMR (CD3OD) 7.44 (d, 1H), 7.32 (t, 1H), 7.05 (d, 1H), 3.56 (m, 1H), 138 (d, 6H). LCMS (m/z): 205.45 (MH)+

Sources & evidence

ORD record
ord-8dd24ca31206472c85acea3ff43aaf54
Source dataset
uspto-grants-2012_12
Patent number
US08338591B2

Reaction notes

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