HCID 5228022, compound → HCID 21962924, compound

HRID 2212005Notes

Reaction equation

HRID 2212005 reaction equation
[Cl:1][C:2]1[CH:3]=[C:4]([CH:14]=[CH:15][C:16]=1[Cl:17])[CH2:5][N:6]1[CH2:11][CH2:10][O:9][CH:8]([CH2:12][NH2:13])[CH2:7]1.[CH3:18][C:19]1[N:23]([C:24]2[CH:29]=[CH:28][CH:27]=[CH:26][CH:25]=2)[N:22]=[CH:21][C:20]=1[CH2:30][C:31](O)=[O:32]>>[Cl:1][C:2]1[CH:3]=[C:4]([CH:14]=[CH:15][C:16]=1[Cl:17])[CH2:5][N:6]1[CH2:11][CH2:10][O:9][CH:8]([CH2:12][NH:13][C:31](=[O:32])[CH2:30][C:20]2[CH:21]=[N:22][N:23]([C:24]3[CH:29]=[CH:28][CH:27]=[CH:26][CH:25]=3)[C:19]=2[CH3:18])[CH2:7]1

Participants

3

Reactant 2

HCID 5228022HCID 5228022, compoundHCID 10308229[4-(3,4-Dichlorobenzyl)morpholin-2-yl]methylamine

Product 1

HCID 21962924HCID 21962924, compound

Procedure

Example 34 was prepared in an analogous manner to Example 1 using a mixture of Intermediate 1 (0.056 g) and (5-methyl-1-phenyl-1H-pyrazol-4-yl)acetic acid (0.0439) to give the title compound (0.014 g).

Workup

  1. customExample 34 was prepared in an analogous manner to Example 1 using

Sources & evidence

ORD record
ord-c2f20c3279ab4743bf01e126129e0461
Source dataset
uspto-grants-2006_09
Patent number
US07101882B2

Reaction notes

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