2,4-Difluoroaniline → HCID 21056591, compound

Participants

Reaction Steps

The title compound was prepared by following the general coupling procedure as a yellow solid (21 mg, 55%) from (4aS,9bR)-bromo-5-methyl-6-trifluoromethyl-1,3,4,4a,5,9b-hexahydro-pyrido[4,3-b]indole-2-carboxylic acid tert-butyl ester (Example 45, 41 mg, 0.095 mmol) and 2,4-difluoroaniline (39 mg, 0.30 mmol). MS (APCI): 384 (base, M+H).

Provenance & Evidence