反应详情

Acylation 8H-Indeno[1,2-d]thiazol-2-ylamine 1b (Prepared in Example 1, Step 2, 377 mg; 2.00 mmol) with 4-pyrazolecarbonyl chloride 12 (208 mg; 1.6 mmol) in a manner similar to that described in Example 7, provided 190 mg of 1H-Pyrazole-4-carboxylic acid (8H-indeno[1,2-d]thiazol-2-yl)-amide 13 as a dark powder.