4-Methoxy-7-morpholinobenzo[d]thiazol-2-amine → HCID 11553749, compound

HRID 2222084Notes

Reaction equation

HRID 2222084 reaction equation
[CH3:1][O:2][C:3]1[C:8]2[N:9]=[C:10]([NH2:12])[S:11][C:7]=2[C:6]([N:13]2[CH2:18][CH2:17][O:16][CH2:15][CH2:14]2)=[CH:5][CH:4]=1.C1([O:25][C:26]([C:28]2[N:29]([CH3:37])[C:30]([CH2:33][N:34]([CH3:36])[CH3:35])=[N:31][CH:32]=2)=O)C=CC=CC=1>>[CH3:1][O:2][C:3]1[C:8]2[N:9]=[C:10]([NH:12][C:26]([C:28]3[N:29]([CH3:37])[C:30]([CH2:33][N:34]([CH3:35])[CH3:36])=[N:31][CH:32]=3)=[O:25])[S:11][C:7]=2[C:6]([N:13]2[CH2:18][CH2:17][O:16][CH2:15][CH2:14]2)=[CH:5][CH:4]=1

Participants

3

Reactant 2

HCID 114028614-Methoxy-7-morpholinobenzo[d]thiazol-2-amineHCID 58592594HCID 58592594, compound

Product 1

HCID 11553749HCID 11553749, compound

Procedure

Using 4-methoxy-7-morpholin-4-yl-benzothiazol-2-ylamine and 2-dimethylaminomethyl-3-methyl-3H-imidazole-4-carboxylic acid phenyl ester, the title compound was obtained as off-white solid (49% yield). MS: m/e=431(M+H+), mp 229-231° C.

Sources & evidence

ORD record
ord-bd4ae857446644b1af529e80114c8719
Source dataset
uspto-grants-2008_05
Patent number
US07371749B2

Reaction notes

Loading…