N-(2-Chloro-5-iodo-pyridin-4-ylmethyl)-N-(4-chloro-2-vinyl-phenyl)-acetamide → 6-Acetyl-3,9-dichloro-5,6-dihydropyrido[4,3-c][1]benzazocine

Participants

Role	Name	HCID	Charge
Reactant	N-(2-Chloro-5-iodo-pyridin-4-ylmethyl)-N-(4-chloro-2-vinyl-phenyl)-acetamide	HCID 59717576	—
Reactant	6-Acetyl-2-chloro-3-fluoro-5,6-dihydro-pyrido[3,2-c][1]benzazocine	HCID 74393412	—
Product	6-Acetyl-3,9-dichloro-5,6-dihydropyrido[4,3-c][1]benzazocine	HCID 72366780	73%

Compound 77C (26 mg, 73%) was prepared from 77B (50 mg, 0.13 mmol) by a route analogous to that used for the preparation of 1D.